, . - ( , ) . , — .
, . 22,5 /3.
— . 0,543 /3.
— . 6 500 000 1 .
— . 49% .
— . , 0,16 .
, - . , .
, . -269 . —
. . .
— . +3420 . .
— (1:1). +4215 .
, . -38,87 . , 13,54 /3.
. - +18° 12140 .
, . 1 0,08988 .
, (. . +17 ). 12,9 /, .. .
, . , .
. 1 50 .
. -40.
. 18--6 .
, . 1990 .
. , , , , 0,005 /3. , .
. 1988 . -, , , –148° . , , – l222u3x.
, . , . 5 , ( ). .
, . (50, ) 0,000026 / . 150 000, Clostridium botulinum.
, . - , .
, 1974 , . , 1300 .
, – , , . 2 .
, , , , 1996 ., «» . : 0,01 ( ) 1 .
, 20 /.
, l- . 100 .
, N-(N-(4-))-2- . 200 000 2% , -
, , . ( ), 3 500 — 6 000 .
, , . 2 .
, , 80- . ( ) 3,7 , 500 .
(). 87,5% . , .
( ). 918 000 000 , .
Chemical Abstracts 1578 . :
Adenosene. N-[4-(dimethylethyl)benzoyl]-2′-O-(tetrahydromethoxypyranyl) adenylyl-(3′→5′)-4-deamino-4-(2,4-dimethylphenoxy)-2′-O-(tetrahydromethoxypyranyl)cytidylyl- (3′→5′)-4-deamino-4-(2,4-dimethylphenoxy)-2′-O-(tetrahydromethoxypyranyl)cytidylyl-(3′→5′)-N- [4-(dimethylethyl)benzoyl]-2′-O-(tetrahydromethoxypyranyl)cytidylyl-(3′→5′)-N-[4-(dimethylethyl) benzoyl]-2′-O-(tetrahydromethoxypyranyl)cytidylyl-(3′→5′)-N-[[4-(dimethylethyl)phenyl]acetyl]-2′-O- (tetrahydromethoxypyranyl)guanylyl-(3′→5′)-N-[[4-(dimethylethyl)phenyl]acetyl]-2′-O- (tetrahydromethoxypyranyl)guanylyl-(3′→5′)-N-[4-(dimethylethyl)benzoyl]-2′-O-(tetrahydromethoxypyranyl) adenylyl-(3′→5′)-N-[4-(dimethylethyl)benzoyl]-2′-O-(tetrahydromethoxypyranyl)cytidylyl-(3′→5′)-4-deamino- 4-(2,4-dimethylphenoxy)-2′-O-(tetrahydromethoxypyranyl)cytidylyl-(3′→5′)-4-deamino-4-(2,4-dimethylphenoxy) -2′-O-(tetrahydromethoxypyranyl)cytidylyl-(3′→5′)-N-[[4-(dimethylethyl)phenyl]acetyl]-2′-O- (tetrahydromethoxypyranyl)guanylyl-(3′→5′)-4-deamino-4-(2,4-dimethylphenoxy)-2′-O-(tetrahydromethoxypyranyl) cytidylyl-(3′→5′)-N-[4-(dimethylethyl)benzoyl]-2′-O-(tetrahydromethoxypyranyl)cytidylyl-(3′→5′)-N-[4- (dimethylethyl)benzoyl]-2′-O-(tetrahydromethoxypyranyl)cytidylyl-(3′→5′)-N-[4-(dimethylethyl)benzoyl] -2′-O-(tetrahydromethoxypyranyl)adenylyl-(3′→5′)-N-[4-(dimethylethyl)benzoyl]-2′-O-(tetrahydromethoxypyranyl) cytidylyl-(3′→5′)-N-[4-(dimethylethyl)benzoyl]-2′-O-(tetrahydromethoxypyranyl)cytidylyl-(3′→5′)-N-[4- (dimethylethyl)benzoyl]-2′,3′-O-(methoxymetylene)-octadecakis(2-chlorophenyl)ester. 5′-[2-(dibromomethyl)benzoate].
16569 . , , 207 000 .
— - , 1840 . ()
— (46,60% )
— (78,09%)
— (90%)
— (10,05 / 0 ), — (0,08929 /)
— (10$ 0,001 )
— 128Te ( 1,5 . 1024 )
- — 148Sm (8 . 1015 )
- — 113Cd (9 . 1015 )
— 5Li (4,4 . 10—22 )
Xe Cs ( 36)
— ( 1 2,4 )
— (. . 3420 )
— ( 320 540 , , , 500-540 )
(97 . 10—6 —1)
— 29SH 49SeH. , ,
— VX (- S-2-() 300 , — 0,3
— TCDD (2,3,7,8--n-), 150000
— d- (LSD) d- (LSD—25)
— R33799 , , 12000
— (10-6 10 $)
, , -269 —